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Researcher
Elise Wouters
Profile
Projects
Publications
Activities
Awards & Distinctions
12
Results
2021
Discovery of a true bivalent dopamine D2 receptor agonist
Mingcheng Qian
Adrián Ricarte
Elise Wouters
James A.R. Dalton
Martijn Risseeuw
Jesús Giraldo
Serge Van Calenbergh
A1
Journal Article
in
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
2021
2020
Assessment of biased agonism among distinct synthetic cannabinoid receptor agonist scaffolds
Elise Wouters
Jolien Walraed
Michael Joseph Robertson
Max Meyrath
Martyna Szpakowska
Andy Chevigné
Georgios Skiniotis
Christophe Stove
A2
Journal Article
in
ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE
2020
Assessment of structure-activity relationships and biased agonism at the Mu opioid receptor of novel synthetic opioids using a novel, stable bio-assay platform
Lakshmi Vasudevan
Marthe Vandeputte
Marie Deventer
Elise Wouters
Annelies Cannaert
Christophe Stove
A1
Journal Article
in
BIOCHEMICAL PHARMACOLOGY
2020
Striatal dopamine D-2-Muscarinic Acetylcholine M-1 Receptor-Receptor interaction in a model of movement disorders
René Crans
Elise Wouters
Marta Valle-Leon
Jaume Taura
Caio M. Massari
Victor Fernandez-Duenas
Christophe Stove
Francisco Ciruela
A1
Journal Article
in
FRONTIERS IN PHARMACOLOGY
2020
2019
Distinct dopamine D2 receptor antagonists differentially impact D2 receptor oligomerization
Elise Wouters
Adrián Ricarte Marín
James Andrew Rupert Dalton
Jesús Giraldo
Christophe Stove
A1
Journal Article
in
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
2019
Functional evaluation of carboxy metabolites of synthetic cannabinoid receptor agonists featuring scaffolds based on L‐valine or L‐tert ‐leucine
Elise Wouters
Lukas Mogler
Annelies Cannaert
Volker Auwärter
Christophe Stove
A1
Journal Article
in
DRUG TESTING AND ANALYSIS
2019
Insights into biased signaling at cannabinoid receptors : synthetic cannabinoid receptor agonists
Elise Wouters
Jolien Walraed
Samuel D. Banister
Christophe Stove
Editorial material
2019
Luminescence- and fluorescence-based complementation assays to screen for GPCR oligomerization : current state of the art
Elise Wouters
Lakshmi Vasudevan
René Crans
Deepak K Saini
Christophe Stove
A1
Journal Article
in
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
2019
The validation of Short Interspersed Nuclear Elements (SINEs) as a RT-qPCR normalization strategy in a rodent model for temporal lobe epilepsy
René Crans
Jana Janssens
Sofie Daelemans
Elise Wouters
Robrecht Raedt
Debby Van Dam
Peter P De Deyn
Kathleen Van Craenenbroeck
Christophe Stove
A1
Journal Article
in
PLOS ONE
2019
Whether it is the action of dopamine or dope : it is all about interaction
Elise Wouters
Christophe Stove
Dissertation
2019
2018
Assessing GPCR dimerization in living cells : comparison of the NanoBiT assay with related bioluminescence- and fluorescence-based approaches
Elise Wouters
Lakshmi Vasudevan
Francisco Ciruela
Deepak Saini
Christophe Stove
Kathleen Van Craenenbroeck
Bookchapter
in
Receptor-receptor interactions in the central nervous system
2018
Synthesis toward bivalent ligands for the dopamine D2 and metabotropic glutamate 5 receptors
Mingcheng Qian
Elise Wouters
James AR Dalton
Martijn Risseeuw
René Crans
Christophe Stove
Jesús Giraldo
Kathleen Van Craenenbroeck
Serge Van Calenbergh
A1
Journal Article
in
JOURNAL OF MEDICINAL CHEMISTRY
2018