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Researcher
Dirk Van Haver
Profile
Projects
Publications
Activities
Awards & Distinctions
40
Results
2009
Development of Analogues of 1 alpha,25-Dihydroxyvitamin D-3 with Biased Side-Chain Orientation: C20 Methylated Des-C,D-homo Analogues
Freek Vrielynck
Dirk Van Haver
Maurits Vandewalle
Lieve Verlinden
Annemieke Verstuyf
Roger Bouillon
Gianluca Croce
Pierre De Clercq
A1
Journal Article
in
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
2009
2007
Mechanism and potential of the growth-inhibitory actions of vitamin D and analogs
G EELEN
C GYSEMANS
L VERLINDEN
E VANOIRBEEK
Pierre De Clercq
Dirk Van Haver
C MATHIEU
R BOUILLON
A VERSTUYF
A1
Journal Article
in
CURRENT MEDICINAL CHEMISTRY
2007
The development of CD-ring modified analogs of 1 alpha,25-dihydroxyvitamin D
Pierre De Clercq
Frederik De Buysser
Garrett Minne
W SCHEPENS
Freek Vrielynck
Dirk Van Haver
M VANDEWALLE
A VERSTUYF
R BOUILLON
A1
Journal Article
in
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY
2007
2006
Asymmetric synthesis of (7aS)-7a-methyl-4,5,7,7a-tetrahydro-1H-indene-2,6-dione and useful derivatives thereof
Samuël Demin
Dirk Van Haver
Pierre De Clercq
A1
Journal Article
in
MOLECULES
2006
Synthesis of spiro[4.5] decane CF-ring analogues of 1 alpha,25-dihydroxyvitamin D-3
Wim Schepens
Dirk Van Haver
Maurits Vandewalle
R BOUILLON
A VERSTUYF
Pierre De Clercq
A1
Journal Article
in
ORGANIC LETTERS
2006
2004
Biological activity and conformational analysis of C20 and C14 epimers of CD-ring modified trans-decalin 1 alpha,25-dihydroxyvitamin D analogs
Pierre De Clercq
Ibrahim Murad
Ling-Jie Gao
Yong-Jun Chen
Dirk Van Haver
Maurits Vandewalle
Annemieke Verstuyf
Lieve Verlinden
Christel Verboven
Roger Bouillon
A1
Journal Article
in
JOURNAL OF STEROID BIOCHEMISTRY AND MOLECULAR BIOLOGY
2004
Synthesis and biological activity of 22-oxa CD-ring modified analogues of 1 α,25-dihydroxyvitamin D3 : cis-perhydrindane CE-ring analogues
Samuël Demin
Dirk Van Haver
Maurits Vandewalle
Pierre De Clercq
R Bouillon
A Verstuyf
A1
Journal Article
in
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
2004
Synthesis and biological activity of 22-oxa CD-ring modified analogues of 1 α,25-dihydroxyvitamin D3 : spiro[5.5]undecane CF-ring analogues
Wim Schepens
Dirk Van Haver
Maurits Vandewalle
Pierre De Clercq
R Bouillon
A Verstuyf
A1
Journal Article
in
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
2004
2003
Previtamin D3 with a trans-fused decalin CD-ring has pronounced genomic activity
L Verlinden
S Verstuyf
C Verboven
G Eelen
C De Ranter
LJ Gao
Y Chen
Ibrahim Murad
M Choi
K Yamamoto
et al.
A1
Journal Article
in
JOURNAL OF BIOLOGICAL CHEMISTRY
2003
Synthesis and binding affinity studies of muscarinic receptor antagonists related to dehydrohimbacine
LJ Gao
Gunther Van Cauwenberge
Noël Hosten
Dirk Van Haver
M Waelbroeck
Pierre De Clercq
A1
Journal Article
in
ARKIVOC
2003
Synthesis, biological activity, and conformational analysis of CD-ring modified trans-decalin 1 alpha,25-dihydroxyvitamin D analogs
YJ CHEN
LJ GAO
Ibrahim Murad
A VERSTUYF
L VERLINDEN
C VERBOVEN
R BOUILLON
D VITERBO
M MILANESIO
Dirk Van Haver
et al.
A1
Journal Article
in
ORGANIC & BIOMOLECULAR CHEMISTRY
2003
2002
A novel short convergent entry into himbacine derivatives
G Van Cauwenberge
LJ Gao
Dirk Van Haver
M Milanesio
D Viterbo
Pierre De Clercq
A1
Journal Article
in
ORGANIC LETTERS
2002
An intramolecular Furan-Diene Diels-Alder approach to 11-oxo 10 alpha-steroids
Sandra Claeys
Dirk Van Haver
Pierre De Clercq
M MILANESIO
D VITERBO
A1
Journal Article
in
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
2002
Evaluation of a two-stage screening procedure in the combinatorial search for serine protease-like activity
Annemieke Madder
L LI
Hilde De Muynck
Nadia Farcy
Dirk Van Haver
Franky Fant
G VANHOENACKER
Patrick Sandra
AP DAVIS
Pierre De Clercq
A1
Journal Article
in
JOURNAL OF COMBINATORIAL CHEMISTRY
2002
Synthesis and affinity studies of himbacine derived muscarinic receptor antagonists
LJ GAO
M WAELBROECK
Sven Hofman
Dirk Van Haver
M MILANESIO
D VITERBO
Pierre De Clercq
A1
Journal Article
in
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
2002
2001
A short intramolecular Diels-Alder route to himbacine derivatives
Sven Hofman
LJ GAO
Hilde Van Dingenen
N HOSTEN
Dirk Van Haver
Pierre De Clercq
M MILANESIO
D VITERBO
A1
Journal Article
in
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
2001
Development of analogues of 1 alpha,25-dihydroxyvitamin D-3 with biased side chain orientation : methylated des-C,D-homo analogues
Stefan Gabriels
Dirk Van Haver
Maurits Vandewalle
Pierre De Clercq
A VERSTUYF
R BOUILLON
A1
Journal Article
in
CHEMISTRY-A EUROPEAN JOURNAL
2001
2000
Biological activity of CD-ring modified 1 alpha,25-dihydroxyvitamin D analogues : C-ring and five-membered D-ring analogues
A VERSTUYF
L VERLINDEN
E VAN ETTEN
L SHI
YS WU
Christiaan D'Halleweyn
Dirk Van Haver
GD ZHU
YJ CHEN
XM ZHOU
et al.
A1
Journal Article
in
JOURNAL OF BONE AND MINERAL RESEARCH
2000
1999
On the unexpected stereochemical outcome of the magnesium in methanol : conjugate reduction of an exocyclic alpha,beta-unsaturated ester
Stefan Gabriels
Dirk Van Haver
Maurits Vandewalle
Pierre De Clercq
Davide Viterbo
A1
Journal Article
in
EUROPEAN JOURNAL OF ORGANIC CHEMISTRY
1999
Synthesis, biological activity, and conformational analysis of four seco-D-15,19-bisnor-1 alpha,25-dihydroxyvitamin D analogues, diastereomeric at C17 and C20
XM ZHOU
GD ZHU
Dirk Van Haver
Maurits Vandewalle
Pierre De Clercq
A VERSTUYF
R BOUILLON
A1
Journal Article
in
JOURNAL OF MEDICINAL CHEMISTRY
1999
1998
On the use of volume maps in the conformational analysis of vitamin D analogs
Dirk Van Haver
Pierre De Clercq
A1
Journal Article
in
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
1998
1997
Mechanism of esterification of 1,3-dimethylamino alcohols by N-acetylimidazole in acetonitrile and the influence of alkyl and geminal dialkyl substitution upon the rate
Annemieke Madder
S SEBASTIAN
Dirk Van Haver
Pierre De Clercq
H MASKILL
A1
Journal Article
in
JOURNAL OF THE CHEMICAL SOCIETY-PERKIN TRANSACTIONS 2
1997
Synthesis of CD-ring modified 1 alpha,25-dihydroxy vitamin D analogues : five-membered D-ring analogues
W Yong
S Ling
Christiaan D'Halleweyn
Dirk Van Haver
Pierre De Clercq
Maurits Vandewalle
A1
Journal Article
in
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
1997
1994
11-fluoro-1-alpha-hydroxyvitamin D-3 : the quest for experimental evidence of the folded vitamin-D conformation
GD ZHU
Dirk Van Haver
H JURRIAANS
Pierre De Clercq
A1
Journal Article
in
TETRAHEDRON
1994
Intramolecular diels-alder reaction of 8-trifluoromethyl-1,3,8-nonatrienes : an access to angular trifluoromethylated hydrindenes
GD ZHU
Bart Van Lancker
Dirk Van Haver
Pierre De Clercq
A1
Journal Article
in
BULLETIN DES SOCIETES CHIMIQUES BELGES
1994
1993
Chemical properties of the natural neurotoxin of Lathyrus sativus 3-N-oxalyl-2,3-diamino-propanoic acid (β-ODAP), its nontoxic 2-N-oxalyl isomer, and its hydrolysis product 2,3-diamino-propanoic acid (DAPRO) by 1H- and 13C-NMR spectroscopy
André De Bruyn
Dirk Van Haver
Fernand Lambein
BM Abegaz
A2
Journal Article
in
NATURAL TOXINS
1993
1992
SYNTHESIS OF (C-11)-SUBSTITUTED ANALOGS OF 1-ALPHA,25-DIHYDROXYVITAMIN-D3.
Christiaan D'Halleweyn
Dirk Van Haver
Johan Van der Eycken
Pierre De Clercq
Maurits Vandewalle
A1
Journal Article
in
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
1992
Synthesis of (C-11)-substituted analogues of 1α,25-dihydroxyvitamin D3
Christiaan D'Halleweyn
Dirk Van Haver
Johan Van der Eycken
Pierre De Clercq
Maurits Vandewalle
A1
Journal Article
in
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS
1992
1989
The synthesis of 4 desoxy-2-azapodophyllotoxins
Johan Van der Eycken
Jean-Paul Bosmans
Dirk Van Haver
Maurits Vandewalle
A Hulkenberg
W Veerman
R Nieuwenhuizen
A1
Journal Article
in
TETRAHEDRON LETTERS
1989
1988
Drug distribution in dog brain studied by positron emission tomography
P Agon
R Braeckman
Dirk Van Haver
H Denutte
P Goethals
H Donche
Franklin Vermeulen
Joris Deman
Jean Kaufman
A1
Journal Article
in
BIOPHARMACEUTICS & DRUG DISPOSITION
1988
1985
Production of C-11-labeled quinidine and tamoxifen
Dirk Van Haver
Tineke Van de Walle
Guido Slegers
Carlo Vandecasteele
A1
Journal Article
in
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
1985
Routine production of 2-deoxy-D-[1-11C]glucose : an alternative
Dirk Van Haver
N.A. Rabi
Maurits Vandewalle
P Goethals
Carlo Vandecasteele
A1
Journal Article
in
JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS
1985
Routine production of H11CN and [11C]-1-Aminocyclopentanecarboxylic acid
JOHAN SAMBRE
Carlo Vandecasteele
Patrick Goethals
N.A. Rabi
Dirk Van Haver
Guido Slegers
A1
Journal Article
in
INTERNATIONAL JOURNAL OF APPLIED RADIATION AND ISOTOPES
1985
1983
Remote-controlled production of 11C-antipyrine
Dirk Van Haver
Pierre De Clercq
Maurits Vandewalle
Tony Vandewalle
Carlo Vandecasteele
C1
Conference
1983
1982
Remote-controlled production of [11C]antipyrine
Dirk Van Haver
Pierre De Clercq
T Van de Walle
C Vandecasteele
A1
Journal Article
in
INTERNATIONAL JOURNAL OF APPLIED RADIATION AND ISOTOPES
1982
1977
1H NMR spectral parameters and configurational assignment of the isomeric 1,4-diacetoxy-2-t-butyl-3-methylcyclopentanes
Dirk Van Haver
M Samson
Maurits Vandewalle
A1
Journal Article
in
TETRAHEDRON
1977
Conformational analysis of prostaglandins F1 based on proton nuclear magnetic resonance spectral data
Pierre De Clercq
M Samson
Dirk Tavernier
Dirk Van Haver
Maurits Vandewalle
A1
Journal Article
in
JOURNAL OF ORGANIC CHEMISTRY
1977
1975
Cyclopentanones : XII. An alternative synthesis of prostaglandins involving catalytic hydrogenation of 2, 3-dialkyl-4-dihydroxy-2-cyclopentenones
R. Coen
Pierre De Clercq
Dirk Van Haver
Maurits Vandewalle
A1
Journal Article
in
BULLETIN DES SOCIÉTÉS CHIMIQUES BELGES
1975
1974
Configurational assignment and 1H-NMR spectral parameters of the isomeric 1,4-diacetoxy-2,3-dimethylcyclopentanes
Dirk Van Haver
Dirk Tavernier
Marc Anteunis
Maurits Vandewalle
A1
Journal Article
in
TETRAHEDRON
1974
Cyclopentanones—VIII : stereochemistry of the lithium-liquid ammonia reduction of 2,3-dialkyl-4-hydroxy-2-cyclopentenones
Pierre De Clercq
Dirk Van Haver
Dirk Tavernier
M Vandewalle
A1
Journal Article
in
TETRAHEDRON
1974